Harnessing Computational & Mechanistic Insights Into Chemoselective Reduction for Engineered Cysteine Site-Specific ADCs

  • Laying out experimental work to develop a novel conjugation method utilizing chemoselective reduction of engineered cysteines, with broad site-specific conjugation applicability
  • Utilizing computational modeling to visualize conjugation sites shielded during circulation
  • Identifying optimized conjugation sites by combining insights from x-ray crystallography structures